Somatostatin Receptor Inhibitors

SSTR1

SSTR2

SSTR3

SSTR5

SSTR4

Somatostatin Receptor Inhibitors, Agonists, Antagonists, Activators, Modulators & Ligands

Nombre del producto	SSTR1	SSTR2	SSTR3	SSTR5	SSTR4	Pureza
Octreotide		SSTR2	SSTR3	SSTR5		99.96%
Cortistatin-14	SSTR1	SSTR2	SSTR3	SSTR5	SSTR4	99.98%
L-797591 hydrochloride	SSTR1					99.81%
SSTR4 agonist 6					SSTR4
CYN 154806		SSTR2				99.97%
Somatostatin-28 (sheep, human rat mouse)				SSTR5		99.67%
Mazisotine					SSTR4, EC₅₀: 4.7 nM	99.54%
CH 275	SSTR1					99.58%
Cyclosomatostatin	SSTR1					99.56%
TT-232	SSTR1				SSTR4	98.72%
NODAGA-LM3		SSTR2				99.65%
BIM-23056			SSTR3	SSTR5		99.98%
Satoreotide		SSTR2				98.80%
CYN 154806 TFA		SSTR2				98.30%
BIM-23190 hydrochloride		SSTR2		SSTR5		99.33%
PRL 2915	hsst₁, Ki: >1000 nM	hsst₂, Ki: 12 nM hsst₂, IC₅₀: 1.8 nM (rat antagonist bioassay versus somatostatin)	hsst₃, Ki: 100 nM	hsst₅, Ki: 520 nM	hsst₄, Ki: 895 nM	99.92%
Veldoreotide TFA		SSTR2, EC₅₀: 37.6 nM	SSTR3, EC₅₀: 31.3 nM		SSTR4, EC₅₀: 10.5 nM	98.97%
Angiopeptin TFA		SSTR2		SSTR5		99.01%
Veldoreotide		SSTR2, EC₅₀: 37.6 nM	SSTR3, EC₅₀: 31.3 nM		SSTR4, EC₅₀: 10.5 nM
Cortistatin-29 (reduced)	SSTR1, IC₅₀: 2.8 nM	SSTR2, IC₅₀: 7.1 nM	SSTR3, IC₅₀: 0.2 nM	SSTR5, IC₅₀: 13.7 nM	SSTR4, IC₅₀: 3.0 nM	98.12%
Seglitide		SSTR2				99.30%
NODAGA-LM3 TFA		SSTR2
PRL 3195	hsst₁, Ki: 1000 nM	hsst₂, Ki: 17 nM	hsst₃, Ki: 66 nM	hsst₅, Ki: 6 nM	hsst₄, Ki: 1000 nM
L-796778			SSTR3			98.00%
Tyr3-Octreotate		SSTR2				99.76%
SSTR3 Agonist-1			SSTR3, EC₅₀: 0.14 nM
[Tyr1]-Somatostatin-14		SSTR2
BN-81674			SSTR3, Ki: 0.92 nM
BIM-23197		SSTR2
SSTR5 antagonist 4				hsst₅, IC₅₀: 1.3 nM
BIM-23056 TFA			SSTR3	SSTR5
SSTR5/TGR5-modulator-1				SSTR5, IC₅₀: 4.37 nM
BIM-23190		SSTR2		SSTR5
Octreotide pamoate		SSTR2	SSTR3	SSTR5
sst2 Receptor agonist-1		SSTR2, Ki: 0.025 nM SSTR2, IC₅₀: 4.8 nM
Cyclosomatostatin TFA	SSTR1
SSTR5 antagonist 7				SSTR5, IC₅₀: 6.2, 25 nM
L803					SSTR4
SSTR4 agonist 5					SSTR4, IC₅₀: 0.228 nM
JR11-PEG3-HBED-CC-PSMA-03		SSTR2
Angiopeptin		SSTR2		SSTR5
Cortistatin-29 (rat)	SSTR1, IC₅₀: 2.8 nM	SSTR2, IC₅₀: 7.1 nM	SSTR3, IC₅₀: 0.2 nM	SSTR5, IC₅₀: 13.7 nM	SSTR4, IC₅₀: 3.0 nM
Onzigolide		SSTR2
SSTR3 agonist-1 TFA			SSTR3, EC₅₀: 0.14 nM
AP102		SSTR2, IC₅₀: 0.63 nM		SSTR5, IC₅₀: 0.65 nM
JR11-PEG3-DOTA-PSMA-03		SSTR2

Name
E-mail *

	Sorry, but the email address you supplied was invalid.